{"id":5902,"date":"2022-02-22T08:09:55","date_gmt":"2022-02-22T08:09:55","guid":{"rendered":"https:\/\/medicinasinc.com\/se\/?post_type=product&#038;p=5902"},"modified":"2022-07-03T23:09:35","modified_gmt":"2022-07-03T23:09:35","slug":"kop-5f-adb","status":"publish","type":"product","link":"https:\/\/medicinasinc.com\/se\/product\/kop-5f-adb\/","title":{"rendered":"K\u00f6p 5F-ADB"},"content":{"rendered":"<p>5F-ADB (alternativt stavat 5F-MDMB-PINACA) \u00e4r en syntetisk cannabinoid som h\u00e4rr\u00f6r fr\u00e5n indazol som har anv\u00e4nts som en aktiv ingrediens i syntetiska cannabisprodukter och s\u00e5lts online som en designerdrog.<\/p>\n<p>5F -ADB \u00e4r en stark agonist av CB1-receptorn, \u00e4ven om dess selektivitet f\u00f6r denna receptor \u00e4r ok\u00e4nd. 5F-ADB hittades f\u00f6r f\u00f6rsta g\u00e5ngen i november 2014 med hj\u00e4lp av obduktionsprov fr\u00e5n en person som dog efter att ha tagit en produkt som inneh\u00e5ller detta l\u00e4kemedel. Efterf\u00f6ljande tester visade att 5F-ADB uppt\u00e4cktes hos totalt tio personer som dog i Japan mellan september och december 2014 av of\u00f6rklarliga drog\u00f6verdoser. Baserat p\u00e5 de relativt l\u00e5ga niv\u00e5erna som uppt\u00e4ckts i v\u00e4vnadstester, anses 5F-ADB vara utomordentligt stark och ser ut att vara betydligt farligare \u00e4n tidigare s\u00e5lda syntetiska cannabisl\u00e4kemedel.<\/p>\n<p>N-[[1-(5- fluorpentyl)-1H-indazol-3-yl]karbonyl]<\/p>\n<p>-3-metyl-D-valinmetylester (5F-ADB) \u00e4r en mycket stark syntetisk cannabis som orsakar sv\u00e5ra psykotiska symtom hos m\u00e4nniskor, ibland d\u00f6dligt.<\/p>\n<p>F\u00f6r att klarg\u00f6ra de neuronala mekanismerna bakom 5F-toxicitet, studerade ADB:s dess effekter p\u00e5 mellanhj\u00e4rnans dopaminerga och serotonerga kretsar, som reglerar en m\u00e4ngd olika grundl\u00e4ggande hj\u00e4rnfunktioner, inklusive de som \u00e4r associerade med bel\u00f6ningsrelaterat beteende. Ex vivo elektrofysiologiska tekniker anv\u00e4ndes f\u00f6r att registrera f\u00f6r\u00e4ndringar i den spontana avfyrningsaktiviteten hos dopaminerga och serotonerga neuroner producerade av 5F-ADB.<\/p>\n<p>5F-ADB (1 M) \u00f6kade dramatiskt den spontana avfyrningshastigheten f\u00f6r dopaminerga neuroner, men misslyckades med att aktivera dem i n\u00e4rvaro av CB1-antagonisten AM251 (1 M). Samma koncentration av 5F-ADB hade \u00e5 andra sidan ingen effekt p\u00e5 serotonerga neuronaktivitet. Dessa fynd visar att 5F-ADB aktiverar lokala CB1-receptorer och f\u00f6rb\u00e4ttrar dopaminerga system i mellanhj\u00e4rnan samtidigt som det inte har n\u00e5gon effekt p\u00e5 serotonerga system i mellanhj\u00e4rnan.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>K\u00f6p 5F-ADB till salu Storbritannien, Europa, Kina (\u00e4ven k\u00e4nd som 5F-MDMB-PINACA) \u00e4r en indazolbaserad syntetisk cannabinoid fr\u00e5n indazol-3-karboxamidfamiljen, tillg\u00e4nglig i grossistledet<\/p>\n","protected":false},"featured_media":5933,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[2596],"product_tag":[4066,4068,4067,4069,4073,4071,4074,4072,4070,4075,4076],"class_list":{"0":"post-5902","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-cannabinoider-till-salu","7":"product_tag-5f-adb","8":"product_tag-5f-adb-pulver","9":"product_tag-5f-adb-till-salu","10":"product_tag-5f-mdmb-pinaca","11":"product_tag-order-5f-adb-online","12":"product_tag-c20h28fn3o3","13":"product_tag-det-bsta-stllet-att-kpa-5f-adb-online","14":"product_tag-how-to-buy-5f-adb-online","15":"product_tag-kp-5f-adb-online","16":"product_tag-v1715016-75-3","17":"product_tag-var-att-kpa-5f-adb-online","19":"first","20":"instock","21":"shipping-taxable","22":"purchasable","23":"product-type-variable"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - 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