{"id":5902,"date":"2022-02-22T08:09:55","date_gmt":"2022-02-22T08:09:55","guid":{"rendered":"https:\/\/medicinasinc.com\/ro\/?post_type=product&#038;p=5902"},"modified":"2022-03-22T00:45:18","modified_gmt":"2022-03-22T00:45:18","slug":"cumpara-5f-adb","status":"publish","type":"product","link":"https:\/\/medicinasinc.com\/ro\/product\/cumpara-5f-adb\/","title":{"rendered":"Cump\u0103ra\u021bi 5F-ADB"},"content":{"rendered":"<p>5F-ADB (scris alternativ 5F-MDMB-PINACA) este un canabinoid sintetic derivat din indazol care a fost utilizat ca ingredient activ \u00een produsele sintetice de canabis \u0219i v\u00e2ndut online ca drog de designer.<\/p>\n<p>5F -ADB este un agonist puternic al receptorului CB1, de\u0219i selectivitatea acestuia pentru acest receptor este necunoscut\u0103. 5F-ADB a fost g\u0103sit pentru prima dat\u0103 \u00een noiembrie 2014 folosind probe post-mortem ob\u021binute de la o persoan\u0103 care a murit dup\u0103 ce a luat un produs care con\u021binea acest medicament. Testele ulterioare au ar\u0103tat c\u0103 5F-ADB a fost detectat la un total de zece persoane care au murit \u00een Japonia \u00eentre septembrie \u0219i decembrie 2014 din cauza supradozelor inexplicabile de droguri. Pe baza nivelurilor relativ sc\u0103zute descoperite \u00een testele tisulare, se crede c\u0103 5F-ADB este extraordinar de puternic \u0219i pare a fi substan\u021bial mai periculos dec\u00e2t medicamentele sintetice de canabis v\u00e2ndute anterior.<\/p>\n<p>N-[[1-(5-). fluoropentil)-1H-indazol-3-il]carbonil]<\/p>\n<p>-3-metil-D-valin\u0103 esterul metilic (5F-ADB) este un canabis sintetic foarte puternic care provoac\u0103 simptome psihotice severe la oameni, ocazional fatal.<\/p>\n<p>Pentru a elucida mecanismele neuronale din spatele toxicit\u0103\u021bii 5F, ADB au studiat efectele acesteia asupra circuitelor dopaminergice \u0219i serotoninergice ale creierului mediu, care regleaz\u0103 o varietate de func\u021bii fundamentale ale creierului, inclusiv cele asociate cu comportamentul legat de recompens\u0103. Tehnicile electrofiziologice ex vivo au fost folosite pentru a \u00eenregistra modific\u0103ri ale activit\u0103\u021bii de declan\u0219are spontan\u0103 a neuronilor dopaminergici \u0219i serotoninergici produ\u0219i de 5F-ADB.<\/p>\n<p>5F-ADB (1 M) a crescut dramatic rata de declan\u0219are spontan\u0103 a neuronilor dopaminergici, dar nu a reu\u0219it s\u0103 le activeze \u00een prezen\u021ba antagonistului CB1 AM251 (1 M). Aceea\u0219i concentra\u021bie de 5F-ADB, pe de alt\u0103 parte, nu a avut niciun efect asupra activit\u0103\u021bii neuronilor serotoninergici. Aceste descoperiri arat\u0103 c\u0103 5F-ADB activeaz\u0103 receptorii locali CB1 \u0219i \u00eembun\u0103t\u0103\u021be\u0219te sistemele dopaminergice din mezencefal, f\u0103r\u0103 a avea niciun efect asupra sistemelor serotoninergice din mezencefal.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Cump\u0103ra\u021bi 5F-ADB de v\u00e2nzare Marea Britanie, Europa, China (cunoscut \u0219i ca 5F-MDMB-PINACA) este un canabinoid sintetic pe baz\u0103 de indazol din familia indazol-3-carboxamide, disponibil\u0103 la comand\u0103 angro<\/p>\n","protected":false},"featured_media":5933,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[2596],"product_tag":[4066,4067,4068,4069,4071,4074,4073,4072,4070,4076,4075],"class_list":{"0":"post-5902","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-canabinoizi-de-vnzare","7":"product_tag-5f-adb","8":"product_tag-5f-adb-de-vanzare","9":"product_tag-5f-adb-pulbere","10":"product_tag-5f-mdmb-pinaca","11":"product_tag-c20h28fn3o3","12":"product_tag-cel-mai-bun-loc-de-cumprare-5f-adb-online","13":"product_tag-comanda-5f-adb-online","14":"product_tag-cum-se-cumpr-5f-adb-online","15":"product_tag-cumpr-5f-adb-online","16":"product_tag-unde-a-cumprare-5f-adb-online","17":"product_tag-v1715016-75-3","19":"first","20":"instock","21":"featured","22":"shipping-taxable","23":"purchasable","24":"product-type-variable"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - 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