{"id":5902,"date":"2022-02-22T08:09:55","date_gmt":"2022-02-22T08:09:55","guid":{"rendered":"https:\/\/medicinasinc.com\/lv\/?post_type=product&#038;p=5902"},"modified":"2022-07-05T22:49:59","modified_gmt":"2022-07-05T22:49:59","slug":"pirkt-5f-adb","status":"publish","type":"product","link":"https:\/\/medicinasinc.com\/lv\/product\/pirkt-5f-adb\/","title":{"rendered":"P\u0113rciet 5F-ADB"},"content":{"rendered":"<p>5F-ADB (alternat\u012bvi rakst\u012bts k\u0101 5F-MDMB-PINACA) ir sint\u0113tisks kanabino\u012bds, kas ieg\u016bts no indazola un ir izmantots k\u0101 akt\u012bv\u0101 sast\u0101vda\u013ca sint\u0113tiskos ka\u0146epju produktos un p\u0101rdots tie\u0161saist\u0113 k\u0101 dizaineru narkotika.<\/p>\n<p>5F -ADB ir sp\u0113c\u012bgs CB1 receptoru agonists, lai gan t\u0101 selektivit\u0101te pret \u0161o receptoru nav zin\u0101ma. 5F-ADB pirmo reizi tika atrasts 2014. gada novembr\u012b, izmantojot p\u0113cn\u0101ves paraugus, kas ieg\u016bti no personas, kura nomira p\u0113c \u0161\u012bs z\u0101les saturo\u0161a produkta lieto\u0161anas. Turpm\u0101kaj\u0101s p\u0101rbaud\u0113s atkl\u0101j\u0101s, ka 5F-ADB tika atkl\u0101ts kopum\u0101 desmit cilv\u0113kiem, kuri Jap\u0101n\u0101 no 2014. gada septembra l\u012bdz decembrim nomira no neizskaidrojamas narkotiku p\u0101rdoz\u0113\u0161anas. Pamatojoties uz sal\u012bdzino\u0161i zemo l\u012bmeni, kas atkl\u0101ts audu p\u0101rbaud\u0113s, tiek uzskat\u012bts, ka 5F-ADB ir \u0101rk\u0101rt\u012bgi sp\u0113c\u012bgs un \u0161\u0137iet daudz b\u012bstam\u0101ks nek\u0101 iepriek\u0161 p\u0101rdot\u0101s sint\u0113tisk\u0101s ka\u0146epju z\u0101les.<\/p>\n<p>N-[[1-(5-) fluoropentil)-1H-indazol-3-il]karbonil]<\/p>\n<p>-3-metil-D-val\u012bna metilesteris (5F-ADB) ir \u013coti sp\u0113c\u012bga sint\u0113tiska ka\u0146epes, kas reiz\u0113m izraisa smagus psihotiskus simptomus cilv\u0113kiem. n\u0101v\u0113jo\u0161s.<\/p>\n<p>Lai noskaidrotu 5F toksicit\u0101tes neironu meh\u0101nismus, m\u0113s p\u0113t\u012bj\u0101m ADB ietekmi uz vidussmadze\u0146u dopam\u012bner\u0123iskaj\u0101m un seroton\u012bner\u0123iskaj\u0101m sh\u0113m\u0101m, kas regul\u0113 da\u017e\u0101das smadze\u0146u pamatfunkcijas, tostarp t\u0101s, kas saist\u012btas ar atalgojuma uzved\u012bbu. Ex vivo elektrofiziolo\u0123isk\u0101s metodes tika izmantotas, lai re\u0123istr\u0113tu 5F-ADB rad\u012bto dopam\u012bner\u0123isko un seroton\u012bner\u0123isko neironu spont\u0101n\u0101s aizdeg\u0161an\u0101s aktivit\u0101tes izmai\u0146as.<\/p>\n<p>5F-ADB (1 M) iev\u0113rojami palielin\u0101ja dopam\u012bner\u0123isko neironu spont\u0101n\u0101s aizdeg\u0161an\u0101s \u0101trumu, bet neizdev\u0101s tos aktiviz\u0113t CB1 antagonista AM251 (1 M) kl\u0101tb\u016btn\u0113. No otras puses, t\u0101da pati 5F-ADB koncentr\u0101cija neietekm\u0113ja seroton\u012bner\u0123isko neironu aktivit\u0101ti. \u0160ie atkl\u0101jumi liecina, ka 5F-ADB aktiviz\u0113 lok\u0101los CB1 receptorus un uzlabo dopam\u012bner\u0123isk\u0101s sist\u0113mas vidussmadzen\u0113s, vienlaikus neietekm\u0113jot seroton\u012bner\u0123isk\u0101s sist\u0113mas vidussmadzen\u0113s.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Ieg\u0101d\u0101jieties 5F-ADB p\u0101rdo\u0161anai Apvienotaj\u0101 Karalist\u0113, Eirop\u0101, \u0136\u012bn\u0101 (paz\u012bstams ar\u012b k\u0101 5F-MDMB-PINACA) ir sint\u0113tisks kanabino\u012bds uz indazola b\u0101zes no indazola-3-karboksam\u012bda saimes, pieejams vairumtirdzniec\u012bb\u0101.<\/p>\n","protected":false},"featured_media":5933,"comment_status":"open","ping_status":"closed","template":"","meta":{"_members_access_role":[],"_members_access_error":""},"product_brand":[],"product_cat":[2596],"product_tag":[4066,4068,4069,4070,4071,4072,4076,4074,4067,4073,4075],"class_list":["post-5902","product","type-product","status-publish","has-post-thumbnail","product_cat-pardodu-kanabinoidus","product_tag-5f-adb","product_tag-5f-adb-pulveris","product_tag-5f-mdmb-pinaca","product_tag-buy-5f-adb-online","product_tag-c20h28fn3o3","product_tag-k-nopirkt-5f-adb-tiesaist","product_tag-kur-nopirkt-5f-adb-tiesaist","product_tag-labk-vieta-kur-iegdties-5f-adb-tiesaist","product_tag-5f-adb-prdoanai","product_tag-pastjums-5f-adb-tiesaist","product_tag-v1715016-75-3","first","instock","shipping-taxable","purchasable","product-type-variable"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v28.0 - 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