{"id":5902,"date":"2022-02-22T08:09:55","date_gmt":"2022-02-22T08:09:55","guid":{"rendered":"https:\/\/medicinasinc.com\/lt\/?post_type=product&#038;p=5902"},"modified":"2022-03-20T12:05:10","modified_gmt":"2022-03-20T12:05:10","slug":"pirkti-5f-adb","status":"publish","type":"product","link":"https:\/\/medicinasinc.com\/lt\/product\/pirkti-5f-adb\/","title":{"rendered":"Pirkite 5F-ADB"},"content":{"rendered":"<p>5F-ADB (kitaip ra\u0161oma 5F-MDMB-PINACA) yra sintetinis kanabinoidas, gautas i\u0161 indazolo, kuris buvo naudojamas kaip aktyvus sintetini\u0173 kanapi\u0173 produkt\u0173 ingredientas ir parduodamas internete kaip dizaineri\u0173 sukurtas narkotikas.<\/p>\n<p>5F -ADB yra stiprus CB1 receptoriaus agonistas, nors jo selektyvumas \u0161iam receptoriui ne\u017einomas. 5F-ADB pirm\u0105 kart\u0105 buvo rastas 2014 m. lapkrit\u012f, naudojant pomirtinius m\u0117ginius, paimtus i\u0161 asmens, mirusio pavartojus \u0161io narkotiko turint\u012f produkt\u0105. V\u0117lesni tyrimai atskleid\u0117, kad 5F-ADB buvo aptiktas i\u0161 viso de\u0161imtyje \u017emoni\u0173, mirusi\u0173 Japonijoje nuo 2014 m. rugs\u0117jo iki gruod\u017eio m\u0117n. nuo nepaai\u0161kinamo narkotik\u0173 perdozavimo. Remiantis santykinai ma\u017eu kiekiu, nustatytu atliekant audini\u0173 tyrimus, manoma, kad 5F-ADB yra nepaprastai stiprus ir atrodo daug pavojingesnis nei anks\u010diau parduoti sintetiniai vaistai nuo kanapi\u0173.<\/p>\n<p>N-[[1-(5-) fluoropentil)-1H-indazol-3-il]karbonil]<\/p>\n<p>-3-metil-D-valino metilo esteris (5F-ADB) yra labai stiprios sintetin\u0117s kanap\u0117s, kartais sukelian\u010dios sunkius psichoz\u0117s simptomus \u017emon\u0117ms. mirtinai.<\/p>\n<p>Siekdami i\u0161siai\u0161kinti 5F toksi\u0161kumo neuroninius mechanizmus, ADB i\u0161tyr\u0117me jo poveik\u012f vidurini\u0173 smegen\u0173 dopaminergin\u0117ms ir serotonergin\u0117ms grandin\u0117ms, kurios reguliuoja \u012fvairias pagrindines smegen\u0173 funkcijas, \u012fskaitant tas, kurios susijusios su elgesiu, susijusiu su atlygiu. Ex vivo elektrofiziologiniai metodai buvo naudojami 5F-ADB gaminam\u0173 dopaminergini\u0173 ir serotonergini\u0173 neuron\u0173 spontaninio u\u017esidegimo poky\u010diams registruoti.<\/p>\n<p>5F-ADB (1 M) smarkiai padidino spontaninio dopaminergini\u0173 neuron\u0173 u\u017edegimo greit\u012f, bet nepavyko j\u0173 suaktyvinti esant CB1 antagonistui AM251 (1 M). Kita vertus, ta pati 5F-ADB koncentracija netur\u0117jo \u012ftakos serotonerginiam neuron\u0173 aktyvumui. \u0160ie radiniai rodo, kad 5F-ADB aktyvuoja vietinius CB1 receptorius ir stiprina dopaminergines sistemas vidurin\u0117se smegenyse, ta\u010diau nedaro jokio poveikio serotonergin\u0117ms sistemoms vidurin\u0117se smegenyse.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Pirkite 5F-ADB pardavimui JK, Europoje, Kinijoje (taip pat \u017einomas kaip 5F-MDMB-PINACA) yra indazolo pagrindu pagamintas sintetinis kanabinoidas i\u0161 indazolo-3-karboksamido \u0161eimos, galimas didmeninis u\u017esakymas<\/p>\n","protected":false},"featured_media":5933,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[2596],"product_tag":[4066,4068,4069,4070,4071,4074,4072,4076,4067,4073,4075],"class_list":{"0":"post-5902","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-parduodami-kanabinoidai","7":"product_tag-5f-adb","8":"product_tag-5f-adb-powder","9":"product_tag-5f-mdmb-pinaca","10":"product_tag-buy-5f-adb-online","11":"product_tag-c20h28fn3o3","12":"product_tag-geriausia-vieta-pirkti-5f-adb-online","13":"product_tag-how-to-buy-5f-adb-online","14":"product_tag-kur-pirkti-5f-adb-online","15":"product_tag-5f-adb-parduodamas","16":"product_tag-u-c5-besisakyti-5f-adb-online","17":"product_tag-v1715016-75-3","19":"first","20":"instock","21":"featured","22":"shipping-taxable","23":"purchasable","24":"product-type-variable"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Pirkite 5F-ADB \u2013 5F-MDMB-PINACA \u2013 geriausius pasaulinius vaistus<\/title>\n<meta name=\"description\" content=\"Pirkite 5F-ADB pardavimui JK, Europa\u00a0(taip pat \u017einomas kaip\u00a05F-MDMB-PINACA) yra indazolo pagrindu pagamintas sintetinis kanabinoidas i\u0161 indazolo-3-karboksamid\u0173 \u0161eimos. 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