{"id":5902,"date":"2022-02-22T08:09:55","date_gmt":"2022-02-22T08:09:55","guid":{"rendered":"https:\/\/medicinasinc.com\/hr\/?post_type=product&#038;p=5902"},"modified":"2022-03-15T05:20:28","modified_gmt":"2022-03-15T05:20:28","slug":"kupiti-5f-adb","status":"publish","type":"product","link":"https:\/\/medicinasinc.com\/hr\/product\/kupiti-5f-adb\/","title":{"rendered":"Kupite 5F-ADB"},"content":{"rendered":"<p>5F-ADB (alternativno napisano 5F-MDMB-PINACA) sintetski je kanabinoid dobiven iz indazola koji se koristio kao aktivni sastojak u proizvodima od sinteti\u010dkog kanabisa i prodaje se online kao dizajnerska droga.<\/p>\n<p>5F. -ADB je jak agonist CB1 receptora, iako je njegova selektivnost za ovaj receptor nepoznata. 5F-ADB je prvi put prona\u0111en u studenom 2014. pomo\u0107u obdukcijskih uzoraka dobivenih od osobe koja je umrla nakon uzimanja proizvoda koji sadr\u017ei ovu drogu. Naknadno testiranje pokazalo je da je 5F-ADB otkriven u ukupno deset ljudi koji su umrli u Japanu izme\u0111u rujna i prosinca 2014. od neobja\u0161njivih predoziranja drogom. Na temelju relativno niskih razina otkrivenih u testovima tkiva, vjeruje se da je 5F-ADB izuzetno jak i izgleda da je znatno opasniji od prethodno prodanih sintetskih lijekova kanabisa.<\/p>\n<p>N-[[1-(5-) fluoropentil)-1H-indazol-3-il]karbonil]<\/p>\n<p>-3-metil-D-valin metil ester (5F-ADB) je vrlo jak sintetski kanabis koji uzrokuje te\u0161ke psihoti\u010dne simptome kod ljudi, povremeno fatalno.<\/p>\n<p>Da bismo razjasnili neuronske mehanizme koji stoje iza 5F-toksi\u010dnosti, ADB-a smo prou\u010davali njegove u\u010dinke na dopaminergi\u010dke i serotonergi\u010dke krugove srednjeg mozga, koji reguliraju niz temeljnih mo\u017edanih funkcija, uklju\u010duju\u0107i one povezane s pona\u0161anjem povezanim s nagradom. Ex vivo elektrofiziolo\u0161ke tehnike kori\u0161tene su za snimanje promjena u spontanoj aktivnosti aktiviranja dopaminergi\u010dkih i serotonergi\u010dkih neurona koje proizvodi 5F-ADB.<\/p>\n<p>5F-ADB (1 M) dramati\u010dno je pove\u0107ao stopu spontanog aktiviranja dopaminergi\u010dkih neurona, ali nije ih uspio aktivirati u prisutnosti CB1 antagonista AM251 (1 M). Ista koncentracija 5F-ADB, s druge strane, nije imala utjecaja na aktivnost serotonergi\u010dkog neurona. Ovi nalazi pokazuju da 5F-ADB aktivira lokalne CB1 receptore i pobolj\u0161ava dopaminergi\u010dke sustave u srednjem mozgu, a da nema utjecaja na serotonergi\u010dke sustave u srednjem mozgu.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Kupite 5F-ADB za prodaju UK, Europa, Kina (tako\u0111er poznat kao 5F-MDMB-PINACA) je sintetski kanabinoid na bazi indazola iz obitelji indazol-3-karboksamida, dostupna je veleprodajna narud\u017eba<\/p>\n","protected":false},"featured_media":5933,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[2596],"product_tag":[4066,4067,4068,4069,4070,4071,4076,4072,4074,4073,4075],"class_list":{"0":"post-5902","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-kanabinoidi-na-prodaju","7":"product_tag-5f-adb","8":"product_tag-5f-adb-za-prodaju","9":"product_tag-5f-adb-prah","10":"product_tag-5f-mdmb-pinaca","11":"product_tag-buy-5f-adb-online","12":"product_tag-c20h28fn3o3","13":"product_tag-gdje-kupiti-5f-adb-online","14":"product_tag-kako-kupiti-5f-adb-online","15":"product_tag-najbolje-mjesto-za-kupnju-5f-adb-online","16":"product_tag-naruiti-5f-adb-online","17":"product_tag-v1715016-75-3","19":"first","20":"instock","21":"featured","22":"shipping-taxable","23":"purchasable","24":"product-type-variable"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - 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